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-Structure paper
Title | The Discovery of a Dual TTK Protein Kinase/CDC2-Like Kinase (CLK2) Inhibitor for the Treatment of Triple Negative Breast Cancer Initiated from a Phenotypic Screen. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 8989-9002, Year 2017 |
Publish date | Sep 27, 2017 (structure data deposition date) |
Authors | Riggs, J.R. / Nagy, M. / Elsner, J. / Erdman, P. / Cashion, D. / Robinson, D. / Harris, R. / Huang, D. / Tehrani, L. / Deyanat-Yazdi, G. ...Riggs, J.R. / Nagy, M. / Elsner, J. / Erdman, P. / Cashion, D. / Robinson, D. / Harris, R. / Huang, D. / Tehrani, L. / Deyanat-Yazdi, G. / Narla, R.K. / Peng, X. / Tran, T. / Barnes, L. / Miller, T. / Katz, J. / Tang, Y. / Chen, M. / Moghaddam, M.F. / Bahmanyar, S. / Pagarigan, B. / Delker, S. / LeBrun, L. / Chamberlain, P.P. / Calabrese, A. / Canan, S.S. / Leftheris, K. / Zhu, D. / Boylan, J.F. |
External links | J. Med. Chem. / PubMed:28991472 |
Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | PDB-6b4w: |
Chemicals | ChemComp-CQ7: ChemComp-CAC: |
Source |
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Keywords | SIGNALING PROTEIN / Protein kinase |