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-Structure paper
Title | Proteome-wide Map of Targets of T790M-EGFR-Directed Covalent Inhibitors. |
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Journal, issue, pages | Cell Chem Biol, Vol. 24, Page 1388-1400.e7, Year 2017 |
Publish date | Feb 21, 2017 (structure data deposition date) |
![]() | Niessen, S. / Dix, M.M. / Barbas, S. / Potter, Z.E. / Lu, S. / Brodsky, O. / Planken, S. / Behenna, D. / Almaden, C. / Gajiwala, K.S. ...Niessen, S. / Dix, M.M. / Barbas, S. / Potter, Z.E. / Lu, S. / Brodsky, O. / Planken, S. / Behenna, D. / Almaden, C. / Gajiwala, K.S. / Ryan, K. / Ferre, R. / Lazear, M.R. / Hayward, M.M. / Kath, J.C. / Cravatt, B.F. |
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Methods | X-ray diffraction |
Resolution | 3.06 Å |
Structure data | ![]() PDB-5uwd: |
Chemicals | ![]() ChemComp-8OV: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / EGFR / kinase / covalent inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |