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-Structure paper
Title | Macrocyclic factor XIa inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 27, Page 4056-4060, Year 2017 |
Publish date | Jun 28, 2017 (structure data deposition date) |
Authors | Wang, C. / Corte, J.R. / Rossi, K.A. / Bozarth, J.M. / Wu, Y. / Sheriff, S. / Myers, J.E. / Luettgen, J.M. / Seiffert, D.A. / Wexler, R.R. / Quan, M.L. |
External links | Bioorg. Med. Chem. Lett. / PubMed:28780160 |
Methods | X-ray diffraction |
Resolution | 2.35 Å |
Structure data | PDB-5wb6: |
Chemicals | ChemComp-9ZM: ChemComp-SO4: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/HYDROLASE inhibitor / HYDROLASE / SERINE PROTEASE / BLOOD COAGULATION FACTOR / PROTEIN INHIBITOR COMPLEX / HYDROLASE-HYDROLASE inhibitor complex |