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Title | Optimization of Allosteric With-No-Lysine (WNK) Kinase Inhibitors and Efficacy in Rodent Hypertension Models. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 7099-7107, Year 2017 |
Publish date | Jul 6, 2017 (structure data deposition date) |
Authors | Yamada, K. / Levell, J. / Yoon, T. / Kohls, D. / Yowe, D. / Rigel, D.F. / Imase, H. / Yuan, J. / Yasoshima, K. / DiPetrillo, K. ...Yamada, K. / Levell, J. / Yoon, T. / Kohls, D. / Yowe, D. / Rigel, D.F. / Imase, H. / Yuan, J. / Yasoshima, K. / DiPetrillo, K. / Monovich, L. / Xu, L. / Zhu, M. / Kato, M. / Jain, M. / Idamakanti, N. / Taslimi, P. / Kawanami, T. / Argikar, U.A. / Kunjathoor, V. / Xie, X. / Yagi, Y.I. / Iwaki, Y. / Robinson, Z. / Park, H.M. |
External links | J. Med. Chem. / PubMed:28771350 |
Methods | X-ray diffraction |
Resolution | 2.006 - 2.458 Å |
Structure data | PDB-5wdy: PDB-5we8: |
Chemicals | ChemComp-ANP: ChemComp-A6S: ChemComp-MN: ChemComp-HOH: ChemComp-A7Y: |
Source |
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Keywords | TRANSFERASE / kinase / inhibitor / TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |