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Title | A 2-Hydroxyisoquinoline-1,3-Dione Active-Site RNase H Inhibitor Binds in Multiple Modes to HIV-1 Reverse Transcriptase. |
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Journal, issue, pages | Antimicrob. Agents Chemother., Vol. 61, Year 2017 |
Publish date | Feb 19, 2017 (structure data deposition date) |
Authors | Kirby, K.A. / Myshakina, N.A. / Christen, M.T. / Chen, Y.L. / Schmidt, H.A. / Huber, A.D. / Xi, Z. / Kim, S. / Rao, R.K. / Kramer, S.T. ...Kirby, K.A. / Myshakina, N.A. / Christen, M.T. / Chen, Y.L. / Schmidt, H.A. / Huber, A.D. / Xi, Z. / Kim, S. / Rao, R.K. / Kramer, S.T. / Yang, Q. / Singh, K. / Parniak, M.A. / Wang, Z. / Ishima, R. / Sarafianos, S.G. |
External links | Antimicrob. Agents Chemother. / PubMed:28760905 |
Methods | X-ray diffraction |
Resolution | 3 Å |
Structure data | PDB-5uv5: |
Chemicals | ChemComp-MN: ChemComp-Y55: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / REVERSE TRANSCRIPTASE / INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |