+Search query
-Structure paper
Title | Discovery of a novel B-cell lymphoma 6 (BCL6)-corepressor interaction inhibitor by utilizing structure-based drug design |
---|---|
Journal, issue, pages | Bioorg. Med. Chem., Vol. 25, Page 4876-4886, Year 2017 |
Publish date | Mar 8, 2017 (structure data deposition date) |
![]() | Yasui, T. / Yamamoto, T. / Sakai, N. / Asano, K. / Takai, T. / Yoshitomi, Y. / Davis, M. / Takagi, T. / Sakamoto, K. / Sogabe, S. ...Yasui, T. / Yamamoto, T. / Sakai, N. / Asano, K. / Takai, T. / Yoshitomi, Y. / Davis, M. / Takagi, T. / Sakamoto, K. / Sogabe, S. / Kamada, Y. / Lane, W. / Snell, G. / Iwata, M. / Goto, M. / Inooka, H. / Sakamoto, J.I. / Nakada, Y. / Imaeda, Y. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.58 - 1.86 Å |
Structure data | ![]() PDB-5x9o: ![]() PDB-5x9p: |
Chemicals | ![]() ChemComp-80R: ![]() ChemComp-EDO: ![]() ChemComp-K: ![]() ChemComp-HOH: ![]() ChemComp-80L: |
Source |
|
![]() | Transcription/Inhibitor / Transcription Repressor / Transcription-Inhibitor complex |