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-Structure paper
Title | Novel Class of Potent and Cellularly Active Inhibitors Devalidates MTH1 as Broad-Spectrum Cancer Target. |
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Journal, issue, pages | ACS Chem. Biol., Vol. 12, Page 1986-1992, Year 2017 |
Publish date | Mar 22, 2017 (structure data deposition date) |
![]() | Ellermann, M. / Eheim, A. / Rahm, F. / Viklund, J. / Guenther, J. / Andersson, M. / Ericsson, U. / Forsblom, R. / Ginman, T. / Lindstrom, J. ...Ellermann, M. / Eheim, A. / Rahm, F. / Viklund, J. / Guenther, J. / Andersson, M. / Ericsson, U. / Forsblom, R. / Ginman, T. / Lindstrom, J. / Silvander, C. / Tresaugues, L. / Giese, A. / Bunse, S. / Neuhaus, R. / Weiske, J. / Quanz, M. / Glasauer, A. / Nowak-Reppel, K. / Bader, B. / Irlbacher, H. / Meyer, H. / Queisser, N. / Bauser, M. / Haegebarth, A. / Gorjanacz, M. |
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Methods | X-ray diffraction |
Resolution | 1.72 Å |
Structure data | ![]() PDB-5nhy: |
Chemicals | ![]() ChemComp-8XT: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / NUDIX / NUCLEOTIDE HYDROLASE / INHIBITOR / ONCOLOGY |