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-Structure paper
Title | JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 8, Page 614-617, Year 2017 |
Publish date | Feb 14, 2017 (structure data deposition date) |
![]() | Newton, A.S. / Deiana, L. / Puleo, D.E. / Cisneros, J.A. / Cutrona, K.J. / Schlessinger, J. / Jorgensen, W.L. |
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Methods | X-ray diffraction |
Resolution | 1.645 - 2 Å |
Structure data | ![]() PDB-5ut4: ![]() PDB-5ut5: ![]() PDB-5ut6: |
Chemicals | ![]() ChemComp-DQX: ![]() ChemComp-GOL: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-2HB: ![]() ChemComp-ACT: ![]() ChemComp-8MY: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Pseudokinase Domain / TRANSFERASE-TRANSFERASE INHIBITOR complex |