+Search query
-Structure paper
Title | Expanding the Scope of Electrophiles Capable of Targeting K-Ras Oncogenes. |
---|---|
Journal, issue, pages | Biochemistry, Vol. 56, Page 3178-3183, Year 2017 |
Publish date | Mar 17, 2017 (structure data deposition date) |
![]() | McGregor, L.M. / Jenkins, M.L. / Kerwin, C. / Burke, J.E. / Shokat, K.M. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.7 - 1.72 Å |
Structure data | ![]() PDB-5v6s: ![]() PDB-5v6v: |
Chemicals | ![]() ChemComp-GDP: ![]() ChemComp-MG: ![]() ChemComp-8YD: ![]() ChemComp-HOH: ![]() ChemComp-CA: ![]() ChemComp-8YA: ![]() ChemComp-GOL: |
Source |
|
![]() | HYDROLASE/HYDROLASE INHIBITOR / K-Ras G12C / covalent inhibitor / HYDROLASE-HYDROLASE INHIBITOR complex |