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-Structure paper
Title | Discovery of a Highly Potent, Cell-Permeable Macrocyclic Peptidomimetic (MM-589) Targeting the WD Repeat Domain 5 Protein (WDR5)-Mixed Lineage Leukemia (MLL) Protein-Protein Interaction. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 4818-4839, Year 2017 |
Publish date | Aug 15, 2012 (structure data deposition date) |
![]() | Karatas, H. / Li, Y. / Liu, L. / Ji, J. / Lee, S. / Chen, Y. / Yang, J. / Huang, L. / Bernard, D. / Xu, J. ...Karatas, H. / Li, Y. / Liu, L. / Ji, J. / Lee, S. / Chen, Y. / Yang, J. / Huang, L. / Bernard, D. / Xu, J. / Townsend, E.C. / Cao, F. / Ran, X. / Li, X. / Wen, B. / Sun, D. / Stuckey, J.A. / Lei, M. / Dou, Y. / Wang, S. |
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Methods | X-ray diffraction |
Resolution | 1.64 - 2.781 Å |
Structure data | ![]() PDB-4gmb: ![]() PDB-5vfc: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-9BA: ![]() ChemComp-SO4: ![]() ChemComp-EDO: |
Source |
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![]() | TRANSCRIPTION/TRANSCRIPTION INHIBITOR / MLL1 / histone methyltransferase / WD40 / TRANSCRIPTION-TRANSCRIPTION INHIBITOR complex / TRANSCRIPTION/INHIBITOR / inhibitor / complex / WD repeat / TRANSCRIPTION / TRANSCRIPTION-INHIBITOR complex |