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Structure paper

Title1,2,4-Triazolo-[1,5-a]pyridine HIF Prolylhydroxylase Domain-1 (PHD-1) Inhibitors With a Novel Monodentate Binding Interaction.
Journal, issue, pagesJ. Med. Chem., Vol. 60, Page 5663-5672, Year 2017
Publish dateMar 1, 2017 (structure data deposition date)
AuthorsAhmed, S. / Ayscough, A. / Barker, G.R. / Canning, H.E. / Davenport, R. / Downham, R. / Harrison, D. / Jenkins, K. / Kinsella, N. / Livermore, D.G. ...Ahmed, S. / Ayscough, A. / Barker, G.R. / Canning, H.E. / Davenport, R. / Downham, R. / Harrison, D. / Jenkins, K. / Kinsella, N. / Livermore, D.G. / Wright, S. / Ivetac, A.D. / Skene, R. / Wilkens, S.J. / Webster, N.A. / Hendrick, A.G.
External linksJ. Med. Chem. / PubMed:28594552
MethodsX-ray diffraction
Resolution2.15 - 2.49 Å
Structure data

PDB-5v18:
Structure of PHD2 in complex with 1,2,4-Triazolo-[1,5-a]pyridine
Method: X-RAY DIFFRACTION / Resolution: 2.15 Å

PDB-5v1b:
Structure of PHD1 in complex with 1,2,4-Triazolo-[1,5-a]pyridine
Method: X-RAY DIFFRACTION / Resolution: 2.49 Å

Chemicals

ChemComp-SO4:
SULFATE ION

ChemComp-8UY:
4-([1,2,4]triazolo[1,5-a]pyridin-5-yl)benzonitrile

ChemComp-FE2:
Unknown entry

ChemComp-HOH:
WATER

ChemComp-FE:
Unknown entry

Source
  • homo sapiens (human)
KeywordsOxidoreductase/Inhibitor / HIF Prolylhydroxylase Domain-2 / Inhibitor / momodentate binding / Oxidoreductase-Inhibitor complex / HIF Prolylhydroxylase Domain-1

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