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Title | A strategy based on nucleotide specificity leads to a subfamily-selective and cell-active inhibitor ofN6-methyladenosine demethylase FTO. |
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Journal, issue, pages | Chem Sci, Vol. 6, Page 112-122, Year 2015 |
Publish date | Apr 9, 2014 (structure data deposition date) |
![]() | Toh, J.D.W. / Sun, L. / Lau, L.Z.M. / Tan, J. / Low, J.J.A. / Tang, C.W.Q. / Cheong, E.J.Y. / Tan, M.J.H. / Chen, Y. / Hong, W. ...Toh, J.D.W. / Sun, L. / Lau, L.Z.M. / Tan, J. / Low, J.J.A. / Tang, C.W.Q. / Cheong, E.J.Y. / Tan, M.J.H. / Chen, Y. / Hong, W. / Gao, Y.G. / Woon, E.C.Y. |
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Methods | X-ray diffraction |
Resolution | 2.65 - 3.1 Å |
Structure data | ![]() PDB-4cxw: ![]() PDB-4cxx: ![]() PDB-4cxy: |
Chemicals | ![]() ChemComp-NI: ![]() ChemComp-6MK: ![]() ChemComp-HOH: ![]() ChemComp-640: ![]() ChemComp-DGR: |
Source |
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![]() | OXIDOREDUCTASE / SMALL MOLECULAR PROBE |