+Search query
-Structure paper
Title | Rational Optimization of Mechanism-Based Inhibitors through Determination of the Microscopic Rate Constants of Inactivation. |
---|---|
Journal, issue, pages | J. Am. Chem. Soc., Vol. 139, Page 7132-7135, Year 2017 |
Publish date | Sep 20, 2016 (structure data deposition date) |
![]() | Eiden, C.G. / Maize, K.M. / Finzel, B.C. / Lipscomb, J.D. / Aldrich, C.C. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | ![]() PDB-5te2: |
Chemicals | ![]() ChemComp-7B9: ![]() ChemComp-PEG: ![]() ChemComp-EDO: ![]() ChemComp-PGE: ![]() ChemComp-HOH: |
Source |
|
![]() | Transferase/Transferase inhibitor / Inhibitor complex / transaminase / PLP / Transferase / Transferase-inhibitor complex / mechanism-based inhibitor / Transferase-Transferase inhibitor complex |