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-Structure paper
Title | 1,4,5-Trisubstituted Imidazole-Based p53-MDM2/MDMX Antagonists with Aliphatic Linkers for Conjugation with Biological Carriers. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 4234-4244, Year 2017 |
Publish date | Apr 6, 2016 (structure data deposition date) |
![]() | Twarda-Clapa, A. / Krzanik, S. / Kubica, K. / Guzik, K. / Labuzek, B. / Neochoritis, C.G. / Khoury, K. / Kowalska, K. / Czub, M. / Dubin, G. ...Twarda-Clapa, A. / Krzanik, S. / Kubica, K. / Guzik, K. / Labuzek, B. / Neochoritis, C.G. / Khoury, K. / Kowalska, K. / Czub, M. / Dubin, G. / Domling, A. / Skalniak, L. / Holak, T.A. |
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Methods | X-ray diffraction |
Resolution | 1.85 - 2 Å |
Structure data | ![]() PDB-5j7f: ![]() PDB-5j7g: |
Chemicals | ![]() ChemComp-6GG: ![]() ChemComp-HOH: |
Source |
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