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-Structure paper
Title | Discovery and Characterization of Novel Nonsubstrate and Substrate NAMPT Inhibitors. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 16, Page 1236-1245, Year 2017 |
Publish date | Nov 30, 2016 (structure data deposition date) |
Authors | Wilsbacher, J.L. / Cheng, M. / Cheng, D. / Trammell, S.A.J. / Shi, Y. / Guo, J. / Koeniger, S.L. / Kovar, P.J. / He, Y. / Selvaraju, S. ...Wilsbacher, J.L. / Cheng, M. / Cheng, D. / Trammell, S.A.J. / Shi, Y. / Guo, J. / Koeniger, S.L. / Kovar, P.J. / He, Y. / Selvaraju, S. / Heyman, H.R. / Sorensen, B.K. / Clark, R.F. / Hansen, T.M. / Longenecker, K.L. / Raich, D. / Korepanova, A.V. / Cepa, S. / Towne, D.L. / Abraham, V.C. / Tang, H. / Richardson, P.L. / McLoughlin, S.M. / Badagnani, I. / Curtin, M.L. / Michaelides, M.R. / Maag, D. / Buchanan, F.G. / Chiang, G.G. / Gao, W. / Rosenberg, S.H. / Brenner, C. / Tse, C. |
External links | Mol. Cancer Ther. / PubMed:28468779 |
Methods | X-ray diffraction |
Resolution | 1.73 - 1.89 Å |
Structure data | PDB-5u2m: PDB-5u2n: |
Chemicals | ChemComp-7T7: ChemComp-SO4: ChemComp-HOH: ChemComp-7TA: |
Source |
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Keywords | Transferase/Transferase Inhibitor / NAMPT inhibitor / Transferase-Transferase Inhibitor complex |