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-Structure paper
Title | Neutral macrocyclic factor VIIa inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 27, Page 2650-2654, Year 2017 |
Publish date | Dec 8, 2016 (structure data deposition date) |
![]() | Wurtz, N.R. / Parkhurst, B.L. / DeLucca, I. / Glunz, P.W. / Jiang, W. / Zhang, X. / Cheney, D.L. / Bozarth, J.M. / Rendina, A.R. / Wei, A. ...Wurtz, N.R. / Parkhurst, B.L. / DeLucca, I. / Glunz, P.W. / Jiang, W. / Zhang, X. / Cheney, D.L. / Bozarth, J.M. / Rendina, A.R. / Wei, A. / Harper, T. / Luettgen, J.M. / Wu, Y. / Wong, P.C. / Seiffert, D.A. / Wexler, R.R. / Priestley, E.S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | ![]() PDB-5u6j: |
Chemicals | ![]() ChemComp-82J: ![]() ChemComp-CA: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / GLYCOPROTEIN / HYDROLASE / SERINE PROTEASE / PLASMA / BLOOD COAGULATION FACTOR / PROTEIN INHIBITOR COMPLEX / CALCIUM- BINDING / HYDROLASE-HYDROLASE INHIBITOR complex |