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TitleSynthesis and biological evaluation of novel selective androgen receptor modulators (SARMs) Part III: Discovery of 4-(5-oxopyrrolidine-1-yl)benzonitrile derivative 2f as a clinical candidate.
Journal, issue, pagesBioorg. Med. Chem., Vol. 25, Page 3330-3349, Year 2017
Publish dateMar 22, 2017 (structure data deposition date)
AuthorsAikawa, K. / Asano, M. / Ono, K. / Habuka, N. / Yano, J. / Wilson, K. / Fujita, H. / Kandori, H. / Hara, T. / Morimoto, M. ...Aikawa, K. / Asano, M. / Ono, K. / Habuka, N. / Yano, J. / Wilson, K. / Fujita, H. / Kandori, H. / Hara, T. / Morimoto, M. / Santou, T. / Yamaoka, M. / Nakayama, M. / Hasuoka, A.
External linksBioorg. Med. Chem. / PubMed:28454849
MethodsX-ray diffraction
Resolution1.44 Å
Structure data

PDB-5v8q:
Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs): Part III
Method: X-RAY DIFFRACTION / Resolution: 1.44 Å

Chemicals

ChemComp-GOL:
GLYCEROL

ChemComp-97A:
4-[(2S,3S)-2-ethyl-3-hydroxy-5-oxopyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsSIGNALING PROTEIN / Androgen Receptor / selective androgen receptor modulators / SARMS

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