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-Structure paper
Title | Virtual screen to NMR (VS2NMR): Discovery of fragment hits for the CBP bromodomain. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 27, Page 2472-2478, Year 2017 |
Publish date | Dec 19, 2016 (structure data deposition date) |
Authors | Spiliotopoulos, D. / Zhu, J. / Wamhoff, E.C. / Deerain, N. / Marchand, J.R. / Aretz, J. / Rademacher, C. / Caflisch, A. |
External links | Bioorg. Med. Chem. Lett. / PubMed:28410781 |
Methods | X-ray diffraction |
Resolution | 1.35 - 1.65 Å |
Structure data | PDB-5mpz: PDB-5mqe: PDB-5mqg: PDB-5mqk: |
Chemicals | ChemComp-4I8: ChemComp-HOH: ChemComp-PKU: ChemComp-F31: ChemComp-QPR: |
Source |
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Keywords | TRANSCRIPTION / CREBBP bromodomain / Inhibitor |