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-Structure paper
Title | Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 27, Page 2003-2009, Year 2017 |
Publish date | Dec 21, 2016 (structure data deposition date) |
![]() | Sun, Z. / Zhang, H. / Chen, Z. / Xie, Y. / Jiang, H. / Chen, L. / Ding, H. / Zhang, Y. / Zheng, M. / Luo, C. |
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Methods | X-ray diffraction |
Resolution | 1.724 Å |
Structure data | ![]() PDB-5wuu: |
Chemicals | ![]() ChemComp-7UU: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / BRD4 / inhibitor / complex |