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-Structure paper
Title | Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells. |
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Journal, issue, pages | Cell Chem Biol, Vol. 24, Page 371-380, Year 2017 |
Publish date | Jun 2, 2015 (structure data deposition date) |
Authors | Tumber, A. / Nuzzi, A. / Hookway, E.S. / Hatch, S.B. / Velupillai, S. / Johansson, C. / Kawamura, A. / Savitsky, P. / Yapp, C. / Szykowska, A. ...Tumber, A. / Nuzzi, A. / Hookway, E.S. / Hatch, S.B. / Velupillai, S. / Johansson, C. / Kawamura, A. / Savitsky, P. / Yapp, C. / Szykowska, A. / Wu, N. / Bountra, C. / Strain-Damerell, C. / Burgess-Brown, N.A. / Ruda, G.F. / Fedorov, O. / Munro, S. / England, K.S. / Nowak, R.P. / Schofield, C.J. / La Thangue, N.B. / Pawlyn, C. / Davies, F. / Morgan, G. / Athanasou, N. / Muller, S. / Oppermann, U. / Brennan, P.E. |
External links | Cell Chem Biol / PubMed:28262558 |
Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | PDB-5a3n: |
Chemicals | ChemComp-ZN: ChemComp-MN: ChemComp-LQT: ChemComp-DMS: ChemComp-PO4: ChemComp-EPE: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE |