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-Structure paper
Title | Dynamic undocking and the quasi-bound state as tools for drug discovery. |
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Journal, issue, pages | Nat Chem, Vol. 9, Page 201-206, Year 2017 |
Publish date | Nov 13, 2015 (structure data deposition date) |
Authors | Ruiz-Carmona, S. / Schmidtke, P. / Luque, F.J. / Baker, L. / Matassova, N. / Davis, B. / Roughley, S. / Murray, J. / Hubbard, R. / Barril, X. |
External links | Nat Chem / PubMed:28221352 |
Methods | X-ray diffraction |
Resolution | 2 - 2.2 Å |
Structure data | PDB-5fnc: PDB-5fnd: PDB-5fnf: |
Chemicals | ChemComp-IEE: ChemComp-SO4: ChemComp-HOH: ChemComp-IQ5: ChemComp-TQL: |
Source |
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Keywords | CHAPERONE / HSP90 / DRUG DESIGN / ONCOLOGY |