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Title | Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 1673-1692, Year 2017 |
Publish date | Jul 7, 2016 (structure data deposition date) |
Authors | Sartori, L. / Mercurio, C. / Amigoni, F. / Cappa, A. / Faga, G. / Fattori, R. / Legnaghi, E. / Ciossani, G. / Mattevi, A. / Meroni, G. ...Sartori, L. / Mercurio, C. / Amigoni, F. / Cappa, A. / Faga, G. / Fattori, R. / Legnaghi, E. / Ciossani, G. / Mattevi, A. / Meroni, G. / Moretti, L. / Cecatiello, V. / Pasqualato, S. / Romussi, A. / Thaler, F. / Trifiro, P. / Villa, M. / Vultaggio, S. / Botrugno, O.A. / Dessanti, P. / Minucci, S. / Zagarri, E. / Carettoni, D. / Iuzzolino, L. / Varasi, M. / Vianello, P. |
External links | J. Med. Chem. / PubMed:28186755 |
Methods | X-ray diffraction |
Resolution | 3.2 Å |
Structure data | PDB-5lgn: |
Chemicals | ChemComp-FAD: ChemComp-6W0: |
Source |
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Keywords | OXIDOREDUCTASE |