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-Structure paper
Title | Targeting Bacillosamine Biosynthesis in Bacterial Pathogens: Development of Inhibitors to a Bacterial Amino-Sugar Acetyltransferase from Campylobacter jejuni. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 2099-2118, Year 2017 |
Publish date | Aug 24, 2016 (structure data deposition date) |
![]() | De Schutter, J.W. / Morrison, J.P. / Morrison, M.J. / Ciulli, A. / Imperiali, B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.94 - 2.1 Å |
Structure data | ![]() PDB-5t2y: ![]() PDB-5tyh: |
Chemicals | ![]() ChemComp-753: ![]() ChemComp-GOL: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-7O4: |
Source |
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![]() | transferase/transferase inhibitor / Campylobacter jejuni bacterial acetyltransferase inhibitor complex / transferase-transferase inhibitor complex / Acetyltransferase Bacterial N-glycan biosynthesis Inhibitor Fragment-based discovery / TRANSFERASE |