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-Structure paper
Title | The juxtamembrane region of TrkA kinase is critical for inhibitor selectivity |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 27, Page 1233-1236, Year 2017 |
Publish date | Oct 26, 2016 (structure data deposition date) |
Authors | Furuya, N. / Momose, T. / Katsuno, K. / Fushimi, N. / Muranaka, H. / Handa, C. / Ozawa, T. / Kinoshita, T. |
External links | Bioorg. Med. Chem. Lett. / PubMed:28159414 |
Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | PDB-5h3q: |
Chemicals | ChemComp-7HF: ChemComp-DTT: ChemComp-NA: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TrkA inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |