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-Structure paper
Title | Allosteric Mutant IDH1 Inhibitors Reveal Mechanisms for IDH1 Mutant and Isoform Selectivity. |
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Journal, issue, pages | Structure, Vol. 25, Page 506-513, Year 2017 |
Publish date | Aug 3, 2016 (structure data deposition date) |
![]() | Xie, X. / Baird, D. / Bowen, K. / Capka, V. / Chen, J. / Chenail, G. / Cho, Y. / Dooley, J. / Farsidjani, A. / Fortin, P. ...Xie, X. / Baird, D. / Bowen, K. / Capka, V. / Chen, J. / Chenail, G. / Cho, Y. / Dooley, J. / Farsidjani, A. / Fortin, P. / Kohls, D. / Kulathila, R. / Lin, F. / McKay, D. / Rodrigues, L. / Sage, D. / Toure, B.B. / van der Plas, S. / Wright, K. / Xu, M. / Yin, H. / Levell, J. / Pagliarini, R.A. |
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Methods | X-ray diffraction |
Resolution | 1.87 - 2.477 Å |
Structure data | ![]() PDB-5sun: ![]() PDB-5svf: ![]() PDB-5svn: ![]() PDB-5svo: |
Chemicals | ![]() ChemComp-NDP: ![]() ChemComp-70Q: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-70P: ![]() ChemComp-FLC: ![]() ChemComp-PEG: ![]() ChemComp-NAP: ![]() ChemComp-EPE: |
Source |
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![]() | OXIDOREDUCTASE / inhibitor / isocitrate dehydrogenase / NADPH / Rossmann fold / MITOCHONDRIAL |