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TitleDiscovery of a Potent, Selective, and Orally Available PI3K delta Inhibitor for the Treatment of Inflammatory Diseases.
Journal, issue, pagesACS Med Chem Lett, Vol. 8, Page 118-123, Year 2017
Publish dateOct 26, 2016 (structure data deposition date)
AuthorsErra, M. / Taltavull, J. / Greco, A. / Bernal, F.J. / Caturla, J.F. / Gracia, J. / Dominguez, M. / Sabate, M. / Paris, S. / Soria, S. ...Erra, M. / Taltavull, J. / Greco, A. / Bernal, F.J. / Caturla, J.F. / Gracia, J. / Dominguez, M. / Sabate, M. / Paris, S. / Soria, S. / Hernandez, B. / Armengol, C. / Cabedo, J. / Bravo, M. / Calama, E. / Miralpeix, M. / Lehner, M.D.
External linksACS Med Chem Lett / PubMed:28105286
MethodsX-ray diffraction
Resolution2.85 Å
Structure data

PDB-5m6u:
HUMAN PI3KDELTA IN COMPLEX WITH LASW1579
Method: X-RAY DIFFRACTION / Resolution: 2.85 Å

Chemicals

ChemComp-7KA:
4-azanyl-6-[[(1~{S})-1-(4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile

Source
  • homo sapiens (human)
KeywordsTRANSFERASE / PI3KDELTA KINASE / PROTEROS BIOSTRUCTURES GMBH

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