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-Structure paper
Title | Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 139, Page 680-685, Year 2017 |
Publish date | May 31, 2016 (structure data deposition date) |
Authors | Zhao, Q. / Ouyang, X. / Wan, X. / Gajiwala, K.S. / Kath, J.C. / Jones, L.H. / Burlingame, A.L. / Taunton, J. |
External links | J. Am. Chem. Soc. / PubMed:28051857 |
Methods | X-ray diffraction |
Resolution | 1.6 - 2.5 Å |
Structure data | PDB-5k9i: PDB-5u8l: |
Chemicals | ChemComp-O44: ChemComp-HOH: ChemComp-SO4: ChemComp-GOL: |
Source |
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Keywords | TRANSFERASE / Covalent Lysine probe / Transferase/Transferase Inhibitor / Kinase Covalent probe Covalent inhibitor Complex / Transferase-Transferase Inhibitor complex |