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-Structure paper
Title | Azaindoles as Zinc-Binding Small-Molecule Inhibitors of the JAMM Protease CSN5. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 56, Page 1294-1297, Year 2017 |
Publish date | Oct 22, 2016 (structure data deposition date) |
Authors | Altmann, E. / Erbel, P. / Renatus, M. / Schaefer, M. / Schlierf, A. / Druet, A. / Kieffer, L. / Sorge, M. / Pfister, K. / Hassiepen, U. ...Altmann, E. / Erbel, P. / Renatus, M. / Schaefer, M. / Schlierf, A. / Druet, A. / Kieffer, L. / Sorge, M. / Pfister, K. / Hassiepen, U. / Jones, M. / Ruedisser, S. / Ostermeier, D. / Martoglio, B. / Jefferson, A.B. / Quancard, J. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:27981705 |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-5m5q: |
Chemicals | ChemComp-ZN: ChemComp-7K1: ChemComp-MPD: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / METAL PROTEASE / COP9 SIGNALOSOME / HYDROXYLASE |