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| Title | Discovery of a PCAF Bromodomain Chemical Probe. |
|---|---|
| Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 56, Page 827-831, Year 2017 |
| Publish date | Oct 21, 2016 (structure data deposition date) |
Authors | Moustakim, M. / Clark, P.G. / Trulli, L. / Fuentes de Arriba, A.L. / Ehebauer, M.T. / Chaikuad, A. / Murphy, E.J. / Mendez-Johnson, J. / Daniels, D. / Hou, C.D. ...Moustakim, M. / Clark, P.G. / Trulli, L. / Fuentes de Arriba, A.L. / Ehebauer, M.T. / Chaikuad, A. / Murphy, E.J. / Mendez-Johnson, J. / Daniels, D. / Hou, C.D. / Lin, Y.H. / Walker, J.R. / Hui, R. / Yang, H. / Dorrell, L. / Rogers, C.M. / Monteiro, O.P. / Fedorov, O. / Huber, K.V. / Knapp, S. / Heer, J. / Dixon, D.J. / Brennan, P.E. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:27966810 |
| Methods | X-ray diffraction |
| Resolution | 2.1 Å |
| Structure data | ![]() PDB-5tpx: |
| Chemicals | ![]() ChemComp-CL: ![]() ChemComp-SO4: ![]() ChemComp-7H7: ![]() ChemComp-HOH: |
| Source |
|
Keywords | TRANSFERASE / Bromodomain / Structural Genomics Consortium (SGC) |
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