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-Structure paper
Title | Sulfonamide-Based Inhibitors of Aminoglycoside Acetyltransferase Eis Abolish Resistance to Kanamycin in Mycobacterium tuberculosis. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 10619-10628, Year 2016 |
Publish date | Mar 18, 2016 (structure data deposition date) |
Authors | Garzan, A. / Willby, M.J. / Green, K.D. / Gajadeera, C.S. / Hou, C. / Tsodikov, O.V. / Posey, J.E. / Garneau-Tsodikova, S. |
External links | J. Med. Chem. / PubMed:27933949 |
Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | PDB-5iv0: |
Chemicals | ChemComp-COA: ChemComp-6E9: ChemComp-CL: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE / Acetyltransferase / Inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |