Structural Characterization and Ligand/Inhibitor Identification Provide Functional Insights into the Mycobacterium tuberculosis Cytochrome P450 CYP126A1.
PDB-5li6: Crystal structure of Mycobacterium tuberculosis CYP126A1 in complex with N-isopropyl-N-((3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl)methyl)-2-(4-nitrophenyl)acetamide 手法: X-RAY DIFFRACTION / 解像度: 1.95 Å
PDB-5li7: Crystal structure of Mycobacterium tuberculosis CYP126A1 in complex with 1-(3-(1H-imidazol-1-yl)propyl)-3-((3s,5s,7s)-adamantan-1-yl)urea 手法: X-RAY DIFFRACTION / 解像度: 1.58 Å
PDB-5li8: Crystal structure of Mycobacterium tuberculosis CYP126A1 in complex with ketoconazole 手法: X-RAY DIFFRACTION / 解像度: 1.83 Å
PDB-5lie: Crystal structure of Mycobacterium tuberculosis CYP126A1 in complex with imidazole 手法: X-RAY DIFFRACTION / 解像度: 1.799 Å