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Structure paper

TitleDiscovery of Indazole Ethers as Novel, Potent, Non-Steroidal Glucocorticoid Receptor Modulators.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 26, Page 5741-, Year 2017
Publish dateJun 8, 2016 (structure data deposition date)
AuthorsHemmerling, M. / Edman, K. / Lepisto, M. / Eriksson, A. / Ivanova, S. / Dahmen, J. / Rehwinkel, H. / Berger, M. / Hendrickx, R. / Dearman, M. ...Hemmerling, M. / Edman, K. / Lepisto, M. / Eriksson, A. / Ivanova, S. / Dahmen, J. / Rehwinkel, H. / Berger, M. / Hendrickx, R. / Dearman, M. / Jensen, T.J. / Wissler, L. / Hansson, T.
External linksBioorg. Med. Chem. Lett. / PubMed:27810243
MethodsX-ray diffraction
Resolution2.2 Å
Structure data

PDB-5g5w:
Structure guided design and discovery of Indazole ethers as highly potent, non-steroidal Glucocorticoid receptor modulators
Method: X-RAY DIFFRACTION / Resolution: 2.2 Å

Chemicals

ChemComp-EDO:
1,2-ETHANEDIOL

ChemComp-R8C:
2,2,2-trifluoro-N-[(1R,2S)-1-{[1-(4-fluorophenyl)-1H-indazol-5-yl]oxy}-1-phenylpropan-2-yl]acetamide

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsHORMONE / GLUCOCORTICOID RECEPTOR / NUCLEAR HORMONE RECEPTOR / STEROID RECEPTOR / SIGNALING PROTEIN / LIGAND COMPLEX / PEPTIDE COMPLEX

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