+Search query
-Structure paper
| Title | Potent Antitumor Activities and Structure Basis of the Chiral beta-Lactam Bridged Analogue of Combretastatin A-4 Binding to Tubulin. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 59, Page 10329-10334, Year 2016 |
| Publish date | Jul 28, 2016 (structure data deposition date) |
Authors | Zhou, P. / Liu, Y. / Zhou, L. / Zhu, K. / Feng, K. / Zhang, H. / Liang, Y. / Jiang, H. / Luo, C. / Liu, M. / Wang, Y. |
External links | J. Med. Chem. / PubMed:27805821 |
| Methods | X-ray diffraction |
| Resolution | 2.48 Å |
| Structure data | ![]() PDB-5gon: |
| Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-GOL: ![]() ChemComp-CA: ![]() ChemComp-GDP: ![]() ChemComp-MES: ![]() ChemComp-6ZR: ![]() ChemComp-IMD: ![]() ChemComp-HOH: |
| Source |
|
Keywords | STRUCTURAL PROTEIN / beta-lactam bridged analogue tubulin colchicine binding site |
Movie
Controller
Structure viewers
About Yorodumi Papers



Authors
External links











Keywords