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-Structure paper
Title | Small-molecule factor D inhibitors targeting the alternative complement pathway. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 12, Page 1105-1110, Year 2016 |
Publish date | Dec 11, 2015 (structure data deposition date) |
Authors | Maibaum, J. / Liao, S.M. / Vulpetti, A. / Ostermann, N. / Randl, S. / Rudisser, S. / Lorthiois, E. / Erbel, P. / Kinzel, B. / Kolb, F.A. ...Maibaum, J. / Liao, S.M. / Vulpetti, A. / Ostermann, N. / Randl, S. / Rudisser, S. / Lorthiois, E. / Erbel, P. / Kinzel, B. / Kolb, F.A. / Barbieri, S. / Wagner, J. / Durand, C. / Fettis, K. / Dussauge, S. / Hughes, N. / Delgado, O. / Hommel, U. / Gould, T. / Mac Sweeney, A. / Gerhartz, B. / Cumin, F. / Flohr, S. / Schubart, A. / Jaffee, B. / Harrison, R. / Risitano, A.M. / Eder, J. / Anderson, K. |
External links | Nat. Chem. Biol. / PubMed:27775713 |
Methods | X-ray diffraction |
Resolution | 1.1 - 1.86 Å |
Structure data | PDB-5fah: PDB-5fbe: PDB-5fbi: PDB-5fck: PDB-5fcr: |
Chemicals | ChemComp-ACT: ChemComp-5VT: ChemComp-HOH: ChemComp-GOL: ChemComp-5W5: ChemComp-5WD: ChemComp-5WC: ChemComp-SO4: ChemComp-EPE: ChemComp-DMS: |
Source |
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Keywords | HYDROLASE |