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| Title | A TPX2 Proteomimetic Has Enhanced Affinity for Aurora-A Due to Hydrocarbon Stapling of a Helix. |
|---|---|
| Journal, issue, pages | ACS Chem. Biol., Vol. 11, Page 3383-3390, Year 2016 |
| Publish date | Sep 22, 2016 (structure data deposition date) |
Authors | Rennie, Y.K. / McIntyre, P.J. / Akindele, T. / Bayliss, R. / Jamieson, A.G. |
External links | ACS Chem. Biol. / PubMed:27775325 |
| Methods | X-ray diffraction |
| Resolution | 2.08 Å |
| Structure data | ![]() PDB-5lxm: |
| Chemicals | ![]() ChemComp-ADP: ![]() ChemComp-PG4: ![]() ChemComp-SO4: ![]() ChemComp-PEG: ![]() ChemComp-MES: ![]() ChemComp-P4G: ![]() ChemComp-CL: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE / Protein kinase / Proteomimetic / Stapled helix peptide / Mitosis |
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homo sapiens (human)
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