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-Structure paper
Title | The Inosine Monophosphate Dehydrogenase, GuaB2, Is a Vulnerable New Bactericidal Drug Target for Tuberculosis. |
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Journal, issue, pages | ACS Infect Dis, Vol. 3, Page 5-17, Year 2017 |
Publish date | Apr 3, 2016 (structure data deposition date) |
Authors | Singh, V. / Donini, S. / Pacitto, A. / Sala, C. / Hartkoorn, R.C. / Dhar, N. / Keri, G. / Ascher, D.B. / Mondesert, G. / Vocat, A. ...Singh, V. / Donini, S. / Pacitto, A. / Sala, C. / Hartkoorn, R.C. / Dhar, N. / Keri, G. / Ascher, D.B. / Mondesert, G. / Vocat, A. / Lupien, A. / Sommer, R. / Vermet, H. / Lagrange, S. / Buechler, J. / Warner, D.F. / McKinney, J.D. / Pato, J. / Cole, S.T. / Blundell, T.L. / Rizzi, M. / Mizrahi, V. |
External links | ACS Infect Dis / PubMed:27726334 |
Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | PDB-5j5r: |
Chemicals | ChemComp-6G1: ChemComp-IMP: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE / inhibitor / IMPDH / mycobacterium / GuaB2 |