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-Structure paper
Title | A New Class of Allosteric HIV-1 Integrase Inhibitors Identified by Crystallographic Fragment Screening of the Catalytic Core Domain. |
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Journal, issue, pages | J. Biol. Chem., Vol. 291, Page 23569-23577, Year 2016 |
Publish date | Jul 7, 2016 (structure data deposition date) |
![]() | Patel, D. / Antwi, J. / Koneru, P.C. / Serrao, E. / Forli, S. / Kessl, J.J. / Feng, L. / Deng, N. / Levy, R.M. / Fuchs, J.R. ...Patel, D. / Antwi, J. / Koneru, P.C. / Serrao, E. / Forli, S. / Kessl, J.J. / Feng, L. / Deng, N. / Levy, R.M. / Fuchs, J.R. / Olson, A.J. / Engelman, A.N. / Bauman, J.D. / Kvaratskhelia, M. / Arnold, E. |
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Methods | X-ray diffraction |
Resolution | 1.651 - 1.7 Å |
Structure data | ![]() PDB-5krs: ![]() PDB-5krt: |
Chemicals | ![]() ChemComp-DMS: ![]() ChemComp-6XI: ![]() ChemComp-HOH: ![]() ChemComp-6W6: |
Source |
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![]() | hydrolase / transferase/inhibitor / HIV-1 Integrase Catalytic Core Domain / p75/LEDGF inhibitor / transferase-inhibitor complex / HIV-1 Integrase; Catalytic Core Domain (CCD); p75/LEDGF inhibitor |