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-Structure paper
Title | A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct. |
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Journal, issue, pages | Oncotarget, Vol. 7, Page 71182-71197, Year 2016 |
Publish date | Aug 9, 2016 (structure data deposition date) |
Authors | Ocasio, C.A. / Rajasekaran, M.B. / Walker, S. / Le Grand, D. / Spencer, J. / Pearl, F.M. / Ward, S.E. / Savic, V. / Pearl, L.H. / Hochegger, H. / Oliver, A.W. |
External links | Oncotarget / PubMed:27563826 |
Methods | X-ray diffraction |
Resolution | 3.1 Å |
Structure data | PDB-5loh: |
Chemicals | ChemComp-STU: ChemComp-CL: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Kinase domain / Inhibitor |