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-Structure paper
Title | First comprehensive structural and biophysical analysis of MAPK13 inhibitors targeting DFG-in and DFG-out binding modes. |
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Journal, issue, pages | Biochim. Biophys. Acta, Vol. 1860, Page 2335-2344, Year 2016 |
Publish date | Nov 3, 2015 (structure data deposition date) |
![]() | Yurtsever, Z. / Patel, D.A. / Kober, D.L. / Su, A. / Miller, C.A. / Romero, A.G. / Holtzman, M.J. / Brett, T.J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2 - 2.594 Å |
Structure data | ![]() PDB-5ekn: ![]() PDB-5eko: |
Chemicals | ![]() ChemComp-N58: ![]() ChemComp-HOH: ![]() ChemComp-N17: |
Source |
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![]() | Transferase/Transferase Inhibitor / KINASE / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX |