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-Structure paper
Title | RVX-297- a novel BD2 selective inhibitor of BET bromodomains. |
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Journal, issue, pages | Biochem. Biophys. Res. Commun., Vol. 477, Page 62-67, Year 2016 |
Publish date | Sep 22, 2015 (structure data deposition date) |
Authors | Kharenko, O.A. / Gesner, E.M. / Patel, R.G. / Norek, K. / White, A. / Fontano, E. / Suto, R.K. / Young, P.R. / McLure, K.G. / Hansen, H.C. |
External links | Biochem. Biophys. Res. Commun. / PubMed:27282480 |
Methods | X-ray diffraction |
Resolution | 1.12 - 1.55 Å |
Structure data | PDB-5dw1: PDB-5dw2: |
Chemicals | ChemComp-5GD: ChemComp-NA: ChemComp-HOH: ChemComp-EDO: |
Source |
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Keywords | PROTEIN BINDING/INHIBITOR / bromodomain / PROTEIN BINDING-INHIBITOR complex |