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-Structure paper
Title | Overcoming EGFR(T790M) and EGFR(C797S) resistance with mutant-selective allosteric inhibitors. |
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Journal, issue, pages | Nature, Vol. 534, Page 129-132, Year 2016 |
Publish date | Aug 7, 2015 (structure data deposition date) |
![]() | Jia, Y. / Yun, C.H. / Park, E. / Ercan, D. / Manuia, M. / Juarez, J. / Xu, C. / Rhee, K. / Chen, T. / Zhang, H. ...Jia, Y. / Yun, C.H. / Park, E. / Ercan, D. / Manuia, M. / Juarez, J. / Xu, C. / Rhee, K. / Chen, T. / Zhang, H. / Palakurthi, S. / Jang, J. / Lelais, G. / DiDonato, M. / Bursulaya, B. / Michellys, P.Y. / Epple, R. / Marsilje, T.H. / McNeill, M. / Lu, W. / Harris, J. / Bender, S. / Wong, K.K. / Janne, P.A. / Eck, M.J. |
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Methods | X-ray diffraction |
Resolution | 2.31 Å |
Structure data | ![]() PDB-5d41: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ANP: ![]() ChemComp-57N: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Allosteric inhibitor / EGFR / TRANSFERASE-TRANSFERASE INHIBITOR complex |