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Title | An inhibitor of KDM5 demethylases reduces survival of drug-tolerant cancer cells. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 12, Page 531-538, Year 2016 |
Publish date | Jul 6, 2015 (structure data deposition date) |
![]() | Vinogradova, M. / Gehling, V.S. / Gustafson, A. / Arora, S. / Tindell, C.A. / Wilson, C. / Williamson, K.E. / Guler, G.D. / Gangurde, P. / Manieri, W. ...Vinogradova, M. / Gehling, V.S. / Gustafson, A. / Arora, S. / Tindell, C.A. / Wilson, C. / Williamson, K.E. / Guler, G.D. / Gangurde, P. / Manieri, W. / Busby, J. / Flynn, E.M. / Lan, F. / Kim, H.J. / Odate, S. / Cochran, A.G. / Liu, Y. / Wongchenko, M. / Yang, Y. / Cheung, T.K. / Maile, T.M. / Lau, T. / Costa, M. / Hegde, G.V. / Jackson, E. / Pitti, R. / Arnott, D. / Bailey, C. / Bellon, S. / Cummings, R.T. / Albrecht, B.K. / Harmange, J.C. / Kiefer, J.R. / Trojer, P. / Classon, M. |
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Methods | X-ray diffraction |
Resolution | 3.14 Å |
Structure data | ![]() PDB-5ceh: |
Chemicals | ![]() ChemComp-NI: ![]() ChemComp-ZN: ![]() ChemComp-50P: ![]() ChemComp-HOH: |
Source |
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![]() | Oxidoreductase/Inhibitor / epigenetics / demethylase / histone / KDM5A / KDM5 / Oxidoreductase-Inhibitor complex |