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Title | Differential Water Thermodynamics Determine Pi3K-Beta/Delta Selectivity for Solvent-Exposed Ligand Modifications. |
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Journal, issue, pages | J. Chem. Inf. Model., Vol. 56, Page 886-, Year 2016 |
Publish date | Sep 16, 2014 (structure data deposition date) |
![]() | Robinson, D. / Bertrand, T. / Carry, J. / Halley, F. / Karlsson, A. / Mathieu, M. / Minoux, H. / Perrin, M. / Robert, B. / Schio, L. / Sherman, W. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.54 Å |
Structure data | ![]() PDB-4v0i: |
Chemicals | ![]() ChemComp-J82: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / PI3K / KINASE SELECTIVITY |