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Title | Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 7, Page 162-166, Year 2016 |
Publish date | Nov 6, 2015 (structure data deposition date) |
Authors | Duncan, K.W. / Rioux, N. / Boriack-Sjodin, P.A. / Munchhof, M.J. / Reiter, L.A. / Majer, C.R. / Jin, L. / Johnston, L.D. / Chan-Penebre, E. / Kuplast, K.G. ...Duncan, K.W. / Rioux, N. / Boriack-Sjodin, P.A. / Munchhof, M.J. / Reiter, L.A. / Majer, C.R. / Jin, L. / Johnston, L.D. / Chan-Penebre, E. / Kuplast, K.G. / Porter Scott, M. / Pollock, R.M. / Waters, N.J. / Smith, J.J. / Moyer, M.P. / Copeland, R.A. / Chesworth, R. |
External links | ACS Med Chem Lett / PubMed:26985292 |
Methods | X-ray diffraction |
Resolution | 2.273 - 2.52 Å |
Structure data | PDB-5emj: PDB-5emk: PDB-5eml: PDB-5emm: |
Chemicals | ChemComp-SFG: ChemComp-5QJ: ChemComp-GOL: ChemComp-HOH: ChemComp-5QH: ChemComp-SAM: ChemComp-5QK: ChemComp-5QL: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / protein-inhibitor complex / TRANSFERASE-TRANSFERASE INHIBITOR complex |