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-Structure paper
Title | Stapled Peptides with gamma-Methylated Hydrocarbon Chains for the Estrogen Receptor/Coactivator Interaction. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 55, Page 4252-4255, Year 2016 |
Publish date | Sep 23, 2015 (structure data deposition date) |
Authors | Speltz, T.E. / Fanning, S.W. / Mayne, C.G. / Fowler, C. / Tajkhorshid, E. / Greene, G.L. / Moore, T.W. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:26928945 |
Methods | X-ray diffraction |
Resolution | 1.5 - 2.271 Å |
Structure data | PDB-5dx3: PDB-5dxb: PDB-5dxe: PDB-5dxg: PDB-5hyr: |
Chemicals | ChemComp-EST: ChemComp-CL: ChemComp-HOH: ChemComp-GOL: |
Source |
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Keywords | Hormone receptor/peptide / Synthetic Peptide / Stapled Peptide / Estrogen Receptor Alpha / Somatic Mutation / Peptide Mimetic / AF-2 Binding / Hormone receptor-peptide complex / Somatic Mutataion / Hormone Receptor / Breast Cancer / Hormone / Estrogen Receptor / GENE REGULATION / Endocrine |