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-Structure paper
Title | Design and Structural Characterization of Potent and Selective Inhibitors of Phosphatidylinositol 4 Kinase III beta. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 1830-1839, Year 2016 |
Publish date | Nov 19, 2015 (structure data deposition date) |
Authors | Rutaganira, F.U. / Fowler, M.L. / McPhail, J.A. / Gelman, M.A. / Nguyen, K. / Xiong, A. / Dornan, G.L. / Tavshanjian, B. / Glenn, J.S. / Shokat, K.M. / Burke, J.E. |
External links | J. Med. Chem. / PubMed:26885694 |
Methods | X-ray diffraction |
Resolution | 3.2 Å |
Structure data | PDB-5euq: |
Chemicals | ChemComp-GDP: ChemComp-SO4: ChemComp-5S8: |
Source |
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Keywords | Transferase/Signaling Protein / lipid kinase / GTPase complex / Transferase-Signaling Protein complex |