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-Structure paper
| Title | SR2067 Reveals a Unique Kinetic and Structural Signature for PPAR gamma Partial Agonism. |
|---|---|
| Journal, issue, pages | Acs Chem. Biol., Vol. 11, Page 273-283, Year 2016 |
| Publish date | Jul 30, 2014 (structure data deposition date) |
Authors | van Marrewijk, L.M. / Polyak, S.W. / Hijnen, M. / Kuruvilla, D. / Chang, M.R. / Shin, Y. / Kamenecka, T.M. / Griffin, P.R. / Bruning, J.B. |
External links | Acs Chem. Biol. / PubMed:26579553 |
| Methods | X-ray diffraction |
| Resolution | 2.22 Å |
| Structure data | ![]() PDB-4r06: |
| Chemicals | ![]() ChemComp-3E7: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
| Source |
|
Keywords | TRANSCRIPTION / nuclear receptor / ligand binding protein |
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homo sapiens (human)
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