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Title | Benzoxazepines Achieve Potent Suppression of IL-17 Release in Human T-Helper 17 (TH 17) Cells through an Induced-Fit Binding Mode to the Nuclear Receptor ROR gamma. |
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Journal, issue, pages | ChemMedChem, Vol. 11, Page 207-216, Year 2016 |
Publish date | Sep 16, 2015 (structure data deposition date) |
![]() | Olsson, R.I. / Xue, Y. / von Berg, S. / Aagaard, A. / McPheat, J. / Hansson, E.L. / Bernstrom, J. / Hansson, P. / Jirholt, J. / Grindebacke, H. ...Olsson, R.I. / Xue, Y. / von Berg, S. / Aagaard, A. / McPheat, J. / Hansson, E.L. / Bernstrom, J. / Hansson, P. / Jirholt, J. / Grindebacke, H. / Leffler, A. / Chen, R. / Xiong, Y. / Ge, H. / Hansson, T.G. / Narjes, F. |
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Methods | X-ray diffraction |
Resolution | 1.54 - 2.1 Å |
Structure data | ![]() PDB-5aph: ![]() PDB-5apj: ![]() PDB-5apk: |
Chemicals | ![]() ChemComp-VYI: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-76E: ![]() ChemComp-NA: |
Source |
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