+Search query
-Structure paper
Title | Potent Inhibitors Active against HIV Reverse Transcriptase with K101P, a Mutation Conferring Rilpivirine Resistance. |
---|---|
Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 1075-1079, Year 2015 |
Publish date | Jun 17, 2015 (structure data deposition date) |
![]() | Gray, W.T. / Frey, K.M. / Laskey, S.B. / Mislak, A.C. / Spasov, K.A. / Lee, W.G. / Bollini, M. / Siliciano, R.F. / Jorgensen, W.L. / Anderson, K.S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 3.5 Å |
Structure data | ![]() PDB-5c42: |
Chemicals | ![]() ChemComp-29T: |
Source |
|
![]() | TRANSFERASE / HYDROLASE/INHIBITOR / HIV / reverse transcriptase / polymerase / non-nucleoside inhibitor / resistance / HYDROLASE-INHIBITOR complex |