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-Structure paper
Title | Structural Basis for Inhibition of Human Autotaxin by Four Potent Compounds with Distinct Modes of Binding. |
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Journal, issue, pages | Mol. Pharmacol., Vol. 88, Page 982-992, Year 2015 |
Publish date | Apr 22, 2015 (structure data deposition date) |
Authors | Stein, A.J. / Bain, G. / Prodanovich, P. / Santini, A.M. / Darlington, J. / Stelzer, N.M. / Sidhu, R.S. / Schaub, J. / Goulet, L. / Lonergan, D. ...Stein, A.J. / Bain, G. / Prodanovich, P. / Santini, A.M. / Darlington, J. / Stelzer, N.M. / Sidhu, R.S. / Schaub, J. / Goulet, L. / Lonergan, D. / Calderon, I. / Evans, J.F. / Hutchinson, J.H. |
External links | Mol. Pharmacol. / PubMed:26371182 |
Methods | X-ray diffraction |
Resolution | 1.75 - 2.95 Å |
Structure data | PDB-4zg6: PDB-4zg7: PDB-4zg9: PDB-4zga: |
Chemicals | ChemComp-ZN: ChemComp-CA: ChemComp-NA: ChemComp-GOL: ChemComp-4NY: ChemComp-SCN: ChemComp-HOH: ChemComp-4O0: ChemComp-NKN: ChemComp-CL: ChemComp-4O2: ChemComp-EDO: ChemComp-ACD: ChemComp-4O3: |
Source |
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Keywords | Hydrolase/Hydrolase Inhibitor / Autotaxin / ENPP2 / inhibitor / Hydrolase-Hydrolase Inhibitor complex |